反应条件
1: 84 percent / K2CO3 / acetone / 5 h / Heating 2: 70 percent / potassium permanganate, pyridine / H2O / 1.) 50 deg C, 3 h, 2.) RT, 3 h View Scheme
参考文献
Claudi, Francesco; Cardellini, Mario; Cingolani, Gian Mario; Piergentili, Alessandro; Pertuzzi, Guidubaldo; Balduini, Walter
Journal of Medicinal Chemistry, 1990 , vol. 33, # 9 p. 2408 - 2412