反应条件
1: n-butyllithium; N,N,N',N,-tetramethylethylenediamine / diethyl ether / 6 h / 0 - 20 °C 2: sodium iodide; AlCl3, aluminium chloride / acetonitrile; dichloromethane / 1 h / 0 - 20 °C View Scheme
参考文献
Rempel, Viktor; Volz, Nicole; Hinz, Sonja; Karcz, Tadeusz; Meliciani, Irene; Nieger, Martin; Wenzel, Wolfgang; Braese, Stefan; Mueller, Christa E.
Journal of Medicinal Chemistry, 2012 , vol. 55, # 18 p. 7967 - 7977