反应条件
1: 88 percent / triethylamine; CH2Cl2 / 2 h / 20 °C 2: 1.) n-BuLi / 1.) THF, hexane, -78 deg C -> 0 deg C, 30 min, 2.) THF, hexane, -78 deg C -> rt, overnight 3: 1.) Li, naphthalene, 2.) H2O / 1.) THF, -78 deg C, 2 h View Scheme
参考文献
Tetrahedron, , vol. 53, # 42 p. 14355 - 14368