反应条件
1: in N,N-dimethyl-formamide
T=25°C; 0.75 h;
2: With potassium carbonate in N,N-dimethyl-formamide
18 h;
参考文献
Marsilje, Thomas H.; Hedrick, Michael P.; Desharnais, Joel; Tavassoli, Ali; Zhang, Yan; Wilson, Ian A.; Benkovic, Stephen J.; Boger, Dale L.
Bioorganic and Medicinal Chemistry, 2003 , vol. 11, # 20 p. 4487 - 4501