1: With BH3*SMe2 in tetrahydrofuran
T=0 - 23°C; 1.95 h;
2: With sodium hydroxide; dihydrogen peroxide in tetrahydrofuran; water
T=23°C; 2 h; Heating / reflux;
参考文献
VICURON PHARMACEUTICALS, INC.
Patent: WO2004/7444 A2, 2004 ;
Location in patent: Page 66 ;