1: With sodium hydride in DMF (N,N-dimethyl-formamide)
T=0 - 70°C; 2.5 h; Heating / reflux;
2: With hydrogenchloride in DMF (N,N-dimethyl-formamide); water
参考文献
VICURON PHARMACEUTICALS, INC.
Patent: WO2004/7444 A2, 2004 ;
Location in patent: Page 95 ;