1: With sodium methylate in tetrahydrofuran; methanol
T=20°C; 3 h; Heating / reflux;
2: With hydrogenchloride in tetrahydrofuran; methanol; water
T=20°C;
参考文献
VICURON PHARMACEUTICALS, INC.
Patent: WO2004/7444 A2, 2004 ;
Location in patent: Page 109 ;