3-氯-n-[4-(1,3-二氧杂烷-2-基)苯基]丙酰胺合成路线 (共 2 条)
反应条件
pyridine in diethyl ether
T=0°C; 0.166667 h;
参考文献
SMITHKLINE BEECHAM CORPORATION
Patent: WO2004/9602 A1, 2004 ;
Location in patent: Page 75 ;
WO 2004/009602 A1
反应条件
N-ethyl-N,N-diisopropylamine in DMF (N,N-dimethyl-formamide)
T=60°C; 4 h;
参考文献
SMITHKLINE BEECHAM CORPORATION
Patent: WO2004/9602 A1, 2004 ;
Location in patent: Page 75-76 ;
WO 2004/009602 A1