甲基4-氰基-2-(乙基氨基)苯甲酸酯合成路线 (共 2 条)
反应条件
trichlorophosphate in pyridine; water
T=20 - 30°C; 1 h;
参考文献
Takeda Pharmaceutical Company Limited
Patent: EP1541576 A1, 2005 ;
Location in patent: Page/Page column 67 ;
EP 1541576 A1
反应条件
sodium tris(acetoxy)borohydride; acetic acid
T=0 - 35°C; 3 h;
参考文献
Takeda Pharmaceutical Company Limited
Patent: EP1568697 A1, 2005 ;
Location in patent: Page/Page column 26 ;