反应条件
palladium diacetate; N-ethyl-N,N-diisopropylamine; tris-(o-tolyl)phosphine in N,N-dimethyl-formamide
T=110°C; Heck reaction; 5 h; Inert atmosphere;
参考文献
Mikami, Satoshi; Kitamura, Shuji; Negoro, Nobuyuki; Sasaki, Shinobu; Suzuki, Masami; Tsujihata, Yoshiyuki; Miyazaki, Takeshi; Ito, Ryo; Suzuki, Nobuhiro; Miyazaki, Junichi; Santou, Takashi; Kanzaki, Naoyuki; Funami, Miyuki; Tanaka, Toshimasa; Yasuma, Tsuneo; Momose, Yu
Journal of Medicinal Chemistry, 2012 , vol. 55, # 8 p. 3756 - 3776