反应条件
1: 88 percent / N,N-diethylaniline, acetic acid / 0.42 h / 190 °C
2: 46 percent / acetic anhydride, acetic acid / 0.58 h / Heating
View Scheme
参考文献
Cowden; Halladay; Cunningham; Hunt; Clark
Journal of Medicinal Chemistry, 1991 , vol. 34, # 6 p. 1818 - 1822