反应条件
1: 50.5 percent / Et3N, DCC / dimethylformamide / 1) DMF, -5 to 0 deg C, 1 h 2) DMF, 5 deg C, overnight
2: NH2OH*HCl, KOH / methanol / Ambient temperature
View Scheme
参考文献
Munakata; Tanaka; Toyoshima
Chemical and Pharmaceutical Bulletin, 1980 , vol. 28, # 7 p. 2045 - 2051
