1: dibenzoyl peroxide; N-bromosuccinmide / tetrachloromethane / 6 h / 100 °C 2: 4-methylmorpholine N-oxide / acetonitrile / 12 h / 20 °C View Scheme
参考文献
BOEHRINGER INGELHEIM INTERNATIONAL GMBH; DE LOMBAERT, Stephane; LIU, Weimin; LO, Ho Yin; NEMOTO, Peter Allen
Patent: WO2012/61169 A1, 2012 ;
WO 2012/061169 A1