反应条件
1: 1.) NaH / 1.) ether, 0 deg C, 1 h, 2.) ether, RT, 8 h
2: 98 percent / H2 / 10 percent Pd/C / aq. ethanol / Ambient temperature
View Scheme
参考文献
Yao, Zhu-Jun; King, Richter C.; Cao, Tin; Kelley, James; Milne, George W. A.; Voigt, Johannes H.; Burke Jr., Terrence R.
Journal of Medicinal Chemistry, 1999 , vol. 42, # 1 p. 25 - 35