2-氨基-5-溴-2,6-二氟苯甲酮合成路线 (共 1 条)
反应条件
1: With zinc(II) chloride
T=120 - 205°C; 3 h;
2: With hydrogenchloride in water
0.5 h; Heating / reflux;
3: With hydrogenchloride in water; acetic acid
T=120°C; 12 h; Heating / reflux;
参考文献
TAKEDA CHEMICAL INDUSTRIES, LTD.
Patent: WO2004/14860 A2, 2004 ;
Location in patent: Page 175-176 ;
WO 2004/014860 A2