反应条件
benzotriazol-1-ol; O-(benzotriazol-1-yl)-N,N,N',N'-tetramethyluronium tetrafluoroborate; N-ethyl-N,N-diisopropylamine in DMF (N,N-dimethyl-formamide)
T=20°C; 24 h;
参考文献
AstraZeneca AB, AstraZeneca AB
Patent: WO2004/16617 A1, 2004 ;
Location in patent: Page 26; 27 ;
WO 2004/016617 A1