反应条件
1: 73 percent / N,N-dimethyl-acetamide / 116 - 118 °C 2: NaOCl, Ac2O, pyridine View Scheme
参考文献
Woo, Peter W. K.; Kostlan, Catherine R.; Sircar, Jagadish C.; Dong, Mi K.; Gilbertsen, Richard B.
Journal of Medicinal Chemistry, 1992 , vol. 35, # 8 p. 1451 - 1457