反应条件
sodium hydride
1.) THF, from 0 deg C to RT, 45 min, 2.) THF, from RT to 60 deg C; Yield given. Multistep reaction;
参考文献
Jones, Terence R.; Webber, Stephen E.; Varney, Michael D.; Reddy, M. Rami; Lewis, Kathleen K.; Kathardekar, Vinit; Mazdiyasni, Hormoz; Deal, Judith; Nguyen, Dzuy; Welsh, Katharine M.; Webber, Stephanie; Johnston, Amanda; Matthews, David A.; Smith, Ward W.; Janson, Cheryl A.; Bacquet, Russell J.; Howland, Eleanor F.; Booth, Carol L. J.; Herrmann, Steven M.; Ward, Robert W.; White, Jennifer; Bartlett, Charlotte A.; Morse, Cathy A.
Journal of Medicinal Chemistry, 1997 , vol. 40, # 5 p. 677 - 683