反应条件
1: sodium hydride / N,N-dimethyl acetamide / 0 °C 2: tris-(dibenzylideneacetone)dipalladium(0); potassium carbonate; 2-(dicyclohexylphosphino)-2',4',6'-tri-i-propyl-1,1’-biphenyl / tert-butyl alcohol / 100 °C View Scheme
参考文献
Deng, Xianming; Yang, Qingkai; Kwiatkowski, Nicholas; Sim, Taebo; McDermott, Ultan; Settleman, Jeffrey E.; Lee, Jiing-Dwan; Gray, Nathanael S.
ACS Medicinal Chemistry Letters, 2011 , vol. 2, # 3 p. 195 - 200