THE GOVERNMENT OF THE UNITED STATES OF AMERICA as represented by THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES 6011
Patent: WO2005/7614 A1, 2005 ;
Location in patent: Page/Page column 36-37; 40-41 ;
WO 2005/007614 A1
1: With N-bromosuccinmide; triethylamine tris(hydrogen fluoride) in dichloromethane
T=0 - 20°C;
2: With potassium tert-butylate in pentane
1 h; Heating;
参考文献
Rosen, Thomas C.; Yoshida, Shinichi; Froehlich, Roland; Kirk, Kenneth L.; Haufe, Guenter
Journal of Medicinal Chemistry, 2004 , vol. 47, # 24 p. 5860 - 5871
