Carter, Percy H.; Cherney, Robert J.; Batt, Douglas G.; Brown, Gregory D.; Duncia, John V.; Gardner, Daniel S.; Yang, Michael G.
Patent: US2005/54626 A1, 2005 ;
Location in patent: Page/Page column 37 ;
US 20050054626 A1
1: 3-tert-butyl-4-methoxybromobenzene With iodine; magnesium in tetrahydrofuran
1 h; Heating / reflux;
2: carbon dioxide in tetrahydrofuran
T=20°C;
3: With hydrogenchloride in tetrahydrofuran; water
参考文献
MEDIVIR AB
Patent: WO2007/144379 A1, 2007 ;
Location in patent: Page/Page column 38 ;