反应条件
1: 85 percent / 1N NaOH / dioxane; methanol / 0 deg C, 5 h, RT
2: 54.6 percent / IBCF, NMMole / dimethylformamide / -20 °C
3: TFA, anisole / CH2Cl2 / 1 h / 0 °C
4: 55 percent
View Scheme
参考文献
Michelot; Mayer; Magneney; Pham Van Chuong; Schmitt; Potier
European Journal of Medicinal Chemistry, 1988 , vol. 23, # 3 p. 243 - 247