3-氯-6-(2-氟-4-甲基-苯基)-吡嗪合成路线 (共 1 条)
反应条件
potassium fluoride; tris-(dibenzylideneacetone)dipalladium(0); tri-tert-butyl phosphine in 1,4-dioxane
T=120°C; 48 h;
参考文献
NOVARTIS AG; NOVARTIS PHARMA GMBH
Patent: WO2004/22556 A1, 2004 ;
Location in patent: Page 23-24 ;
WO 2004/022556 A1