1: 3,5-dimethyl-1H-pyrazole With potassium hydroxide in dimethyl sulfoxide
T=80°C; 1 h; Inert atmosphere;
2: benzyl chloride in dimethyl sulfoxide
T=20°C; 2 h; Inert atmosphere;
参考文献
Chavez, Sherry A.; Martinko, Alexander J.; Lau, Corinna; Pham, Michael N.; Cheng, Kui; Bevan, Douglas E.; Mollnes, Tom E.; Yin, Hang
Journal of Medicinal Chemistry, 2011 , vol. 54, # 13 p. 4659 - 4669