5-氯-2,3-二氢-1H-茚-1-胺合成路线 (共 2 条)
反应条件
1: With ammonium acetate in isopropyl alcohol T=20°C; 1 h; 2: With sodium cyanoborohydride in isopropyl alcohol 2 h; Heating; Further stages.;
参考文献
Journal of Medicinal Chemistry, , vol. 51, # 3 p. 392 - 395
反应条件
ammonium chloride; acetic acid; zinc T=30°C; 24 h;
参考文献
WO2012/135166 A1, ;
Page/Page column 78 ;
WO 2012/135166 A1