反应条件
1: 86 percent / POCl3 / benzene / 2 h / Heating 2: 89 percent / HCO2H; Et3N / (S,S)-TsDPEN-Ru(II) complex / dimethylformamide / 12 h / 20 °C 3: 78 percent / AlH3 / tetrahydrofuran / 0.17 h / 20 °C 4: 98 percent / SOCl2 / 0 - 20 °C View Scheme
参考文献
Santos, Leonardo S.; Pilli, Ronaldo A.; Rawal, Viresh H.
Journal of Organic Chemistry, 2004 , vol. 69, # 4 p. 1283 - 1289