1: C7H8O3S*C12H21NO2; di-tert-butyl dicarbonate With sodium hydroxide in tetrahydrofuran; water T=10 - 17°C; 2 h; 2: tert-butylamine With sodium hydroxide in tetrahydrofuran; water T=0 - 20°C; pH=12; 3: With hydrogenchloride in water
参考文献
MERCK and CO., INC.
Patent: WO2004/24720 A1, 2004 ;
Location in patent: Page 73 ;
WO 2004/024720 A1