反应条件
1: phosphorus pentachloride / chloroform / 3.25 h / 0 °C / |Reflux
2: lithium carbonate / N,N-dimethyl-formamide / 7 h / 120 °C
3: lithium carbonate / N,N-dimethyl-formamide / 3 h / 130 °C
View Scheme
参考文献
Wu, Yuelin; Min, Xiao; Zhuang, Chunlin; Li, Jin; Yu, Zhiliang; Dong, Guoqiang; Yao, Jiangzhong; Wang, Shengzheng; Liu, Yang; Wu, Shanchao; Zhu, Shiping; Sheng, Chunquan; Wei, Yunyang; Zhang, Huojun; Zhang, Wannian; Miao, Zhenyuan
European Journal of Medicinal Chemistry, 2014 , vol. 82, p. 545 - 551