5-溴-1,2-苯并异噻唑-3-甲酸合成路线 (共 2 条)
反应条件
sulfuric acid; bromine; nitric acid; acetic acid T=70°C;
参考文献
ACS Medicinal Chemistry Letters, , vol. 1, # 1 p. 19 - 23
参考文献
MEMORY PHARMACEUTICALS CORPORATION
Patent: WO2007/56582 A1, 2007 ;
Location in patent: Page/Page column 69 ;
WO 2007/056582 A1