N-丙-2-炔基吡啶-4-甲酰胺合成路线 (共 1 条)
反应条件
benzotriazol-1-ol; 1-ethyl-(3-(3-dimethylamino)propyl)-carbodiimide hydrochloride; triethylamine in N,N-dimethyl-formamide
T=20°C; 48 h;
参考文献
Zhang, Jianjun; Chiang, Fang-I.; Wu, Long; Czyryca, Przemyslaw Greg; Li, Ding; Chang, Cheng-Wei Tom
Journal of Medicinal Chemistry, 2008 , vol. 51, # 23 p. 7563 - 7573