反应条件
1: 7-CHLORO-3-(4-METHOXYPHENYL)-1H-INDAZOLE With sodium hydride in N,N-dimethyl-formamide
2: propyl halide in N,N-dimethyl-formamide
T=60°C;
3: With boron tribromide in dichloromethane; cyclohexane
T=20°C; 5 h;
参考文献
Steffan, Robert J.; Matelan, Edward; Ashwell, Mark A.; Moore, William J.; Solvibile, William R.; Trybulski, Eugene; Chadwick, Christopher C.; Chippari, Susan; Kenney, Thomas; Eckert, Amy; Borges-Marcucci, Lisa; Keith, James C.; Xu, Zhang; Mosyak, Lydia; Harnish, Douglas C.
Journal of Medicinal Chemistry, 2004 , vol. 47, # 26 p. 6435 - 6438
