1-[1-(4-吡啶基)环丙基]甲胺合成路线 (共 1 条)
反应条件
1: With sodium hydroxide; phenylmethyltriethylammonium bromide in water
T=20 - 50°C; 4.25 h;
2: With ammonia; hydrogen; nickel in methanol; water
P=2585.81 Torr;
参考文献
ELIAN PHARMACEUTICALS INC
Patent: WO2004/33436 A1, 2004 ;
Location in patent: Page 69 ;
WO 2004/033436 A1