1-(4-三氟甲基苯基)哌啶-4-醇合成路线 (共 1 条)
反应条件
sodium t-butanolate; tris-(dibenzylideneacetone)dipalladium(0); 2,2'-bis-(diphenylphosphino)-1,1'- binaphthyl in toluene T=120°C; 1 h; Microwave irradiation;
参考文献
SHIONOGI and CO., LTD.
Patent: EP1988077 A1, 2008 ;
Location in patent: Page/Page column 63-64 ;