1.1: sulfuric acid / 72 h / |Reflux 2.1: N-bromosuccinmide; 2,2'-azo-bisisobutyronitrile / benzene / 80 °C 3.1: ammonia / methanol / 20 °C 4.1: sodium hydride / N,N-dimethyl-formamide / 0.5 h / 0 °C / |Inert atmosphere 4.2: 1 h / 20 °C / |Inert atmosphere View Scheme
参考文献
PETER MACCALLUM CANCER INSTITUTE; SPICER, Julie Ann; DENNY, William Alexander; MILLER, Christian Karl; O'CONNOR, Patrick David; HUTTUNEN, Kristiina; TRAPANI, Joseph A.; HILL, Geoff; ALEXANDER, Kylie
Patent: WO2014/28968 A1, 2014 ;