反应条件
2,2,6,6-tetramethyl-piperidine; n-butyllithium in tetrahydrofuran
T=-78 - 20°C; Inert atmosphere;
参考文献
QUANTICEL PHARMACEUTICALS, INC; NIE, Zhe; STAFFORD, Jeffrey, Alan; VEAL, James, Marvin; WALLACE, Michael, Brennan
Patent: WO2014/89364 A1, 2014 ;
Location in patent: Paragraph 00896; 00897 ;