反应条件
1: 98 percent / 12N HCl, H2 / 10percent Pd/C / methanol / 25 °C / 2068.6 - 2327.2 Torr
2: ICl, 4N aq. HCl / 18 h / 20 - 25 °C
View Scheme
参考文献
Stokker; Smith; Cragoe Jr.; Ludden; Russo; Sweet; Watson
Journal of Medicinal Chemistry, 1981 , vol. 24, # 1 p. 115 - 117