1,2,3,6-四氢吡啶合成路线

参考文献

Hu, X.Eric; Kim, Nick K; Ledoussal, Benoit; Colson, Anny-Odile
Tetrahedron Letters, 2002 , vol. 43, # 23 p. 4289 - 4293

参考文献

BRISTOL-MYERS SQUIBB COMPANY
Patent: WO2005/66176 A1, 2005 ;
Location in patent: Page/Page column 62-63 ;
WO 2005/066176 A1

694-05-31,2,3,6-四氢吡啶+

1885-14-9氯甲酸苯酯

66207-23-6N-苯甲氧基甲酰基-1,2,5,6-四氢吡啶

参考文献

Zeneca Limited
Patent: US5654299 A1, 1997 ;

694-05-31,2,3,6-四氢吡啶+

75315-63-82,5-二氧代吡咯烷-1-羧酸苄酯

66207-23-6N-苯甲氧基甲酰基-1,2,5,6-四氢吡啶

参考文献

Newhouse, Bradley J.; Hansen, Joshua D.; Grina, Jonas; Welch, Mike; Topalov, George; Littman, Nicole; Callejo, Michele; Martinson, Matthew; Galbraith, Sarah; Laird, Ellen R.; Brandhuber, Barbara J.; Vigers, Guy; Morales, Tony; Woessner, Rich; Randolph, Nikole; Lyssikatos, Joseph; Olivero, Alan
Bioorganic and Medicinal Chemistry Letters, 2011 , vol. 21, # 11 p. 3488 - 3492

694-05-31,2,3,6-四氢吡啶+

108-90-7氯苯

26905-02-24-(4-氯苯基)哌啶+

100129-35-94-(2-氯苯基)哌啶+

99329-53-04-(3-氯苯基l)-哌啶

参考文献

Klumpp, Douglas A.; Beauchamp, Philip S.; Sanchez Jr., Gregorio V.; Aguirre, Sharon; De Leon, Sarah
Tetrahedron Letters, 2001 , vol. 42, # 34 p. 5821 - 5823

694-05-31,2,3,6-四氢吡啶+

462-06-6氟苯

37656-48-74-(4-氟苯基)呱碇+

104774-88-14-(3-氟苯基)哌啶+

180161-17-54-(2-氟苯基)哌啶

参考文献

Tetrahedron Letters, , vol. 42, # 34 p. 5821 - 5823

694-05-31,2,3,6-四氢吡啶+

462-06-6氟苯

37656-48-74-(4-氟苯基)呱碇+

104774-88-14-(3-氟苯基)哌啶+

180161-17-54-(2-氟苯基)哌啶

参考文献

Klumpp, Douglas A.; Beauchamp, Philip S.; Sanchez Jr., Gregorio V.; Aguirre, Sharon; De Leon, Sarah
Tetrahedron Letters, 2001 , vol. 42, # 34 p. 5821 - 5823

694-05-31,2,3,6-四氢吡啶+

108-88-3甲苯

59083-39-54-(4-甲基苯基)哌啶+

111153-83-4+

630116-52-84-(2-甲苯基)哌啶

参考文献

Klumpp, Douglas A.; Beauchamp, Philip S.; Sanchez Jr., Gregorio V.; Aguirre, Sharon; De Leon, Sarah
Tetrahedron Letters, 2001 , vol. 42, # 34 p. 5821 - 5823

694-05-31,2,3,6-四氢吡啶+

10443-65-92-溴丙烯酸

139021-47-9

参考文献

Grigg; Santhakumar; Sridharan; Stevenson; Teasdale; Thornton-Pett; Worakun
Tetrahedron, 1991 , vol. 47, # 46 p. 9703 - 9720

694-05-31,2,3,6-四氢吡啶+

24424-99-5二碳酸二叔丁酯

161157-50-27-氧杂-3-氮杂双环[4.1.0]庚烷-3-羧酸叔丁酯

参考文献

Robin, Aelig; Koehler, Valentin; Jones, Alison; Ali, Afruja; Kelly, Paul P.; O'Reilly, Elaine; Turner, Nicholas J.; Flitsch, Sabine L.
Beilstein Journal of Organic Chemistry, 2011 , vol. 7, art. no. 7, p. 1494 - 1498