反应条件
1: With 2,2,6,6-tetramethyl-piperidine; n-butyllithium; N,N,N',N,-tetramethylethylenediamine; zinc(II) chloride in tetrahydrofuran
T=0 - 20°C; 2 h;
2: With iodine in tetrahydrofuran
16 h;
参考文献
Nguyen, Thi Thanh Binh; Lomberget, Thierry; Tran, Ngoc Chau; Colomb, Evelyne; Nachtergaele, Lore; Thoret, Sylviane; Dubois, Joelle; Guillaume, Joren; Abdayem, Rawad; Haftek, Marek; Barret, Roland
Bioorganic and Medicinal Chemistry Letters, 2012 , vol. 22, # 23 p. 7227 - 7231