反应条件
1: 79 percent / triethylamine / dimethylformamide 2: 100 percent / DMF*SO3 / dimethylformamide; pyridine / 2 h / 30 °C / other reagent (Pyr*SO3) 3: 66 percent / AcOH, H2 / Pd/C (5percent) / dimethylformamide; methanol / 2 h / Ambient temperature View Scheme
参考文献
Futaki, Shiroh; Taike, Takashi; Yagami, Takeshi; Ogawa, Toyoko; Akita, Tadashi; Kitagawa, Kouki
Journal of the Chemical Society, Perkin Transactions 1: Organic and Bio-Organic Chemistry (1972-1999), 1990 , p. 1739 - 1744