反应条件
1: N-(9-fluorenylmethoxycarbonyl)glycine With benzotriazol-1-ol; O-(1H-benzotriazol-1-yl)-N,N,N',N'-tetramethyluronium hexafluorophosphate; N-ethyl-N,N-diisopropylamine in N,N-dimethyl-formamide Wang resin; Automated synthesizer; 2: With piperidine in 1-methyl-pyrrolidin-2-one Wang resin; Automated synthesizer; 3: 9-fluorenylmethyloxycarbonyl-Cys-OH; protected (S)-2-aminopentanedioic acid Further stages;
参考文献
Tetrahedron, , vol. 69, # 52 p. 11130 - 11137
