反应条件
1: 90 percent / HOBt*H2O, NEt3, DCC / dimethylformamide / a) -5 deg C to 0 deg C, 1 h, b) 20 deg C, 24 h 2: 86 percent / 0.5 M NaOH / acetone / 1.5 h 3: 90 percent / 1.3 M HCl/AcOH / 1 h View Scheme
参考文献
Smith, D. David; Boyd, Kenneth G.; Hopton, David; Baxter, Robert L.; Ramage, Robert
Journal of the Chemical Society, Perkin Transactions 1: Organic and Bio-Organic Chemistry (1972-1999), 1993 , # 5 p. 551 - 556