1-乙酰基-3,2-甲苯甲酰基-5-氟尿嘧啶合成路线 (共 2 条)
反应条件
triethylamine in 1,4-dioxane
1.5 h; Ambient temperature;
参考文献
Kametani, Tetsuji; Kigasawa, Kazuo; Hiiragi, Mineharu; Wakisaka, Kikuo; Haga, Seiji; et al.
Journal of Medicinal Chemistry, 1980 , vol. 23, # 12 p. 1324 - 1329
反应条件
pyridine in 1,4-dioxane
T=80°C; 2 h;
参考文献
Kametani, Tetsuji; Kigasawa, Kazuo; Hiiragi, Mineharu; Wakisaka, Kikuo; Haga, Seiji; et al.
Journal of Medicinal Chemistry, 1980 , vol. 23, # 12 p. 1324 - 1329