1-[3-(三氟甲基)苯基]-4-羟基哌啶合成路线 (共 1 条)
反应条件
potassium carbonate; sodium iodide in N,N-dimethyl-formamide
T=100°C; Alkylation; Cyclization;
参考文献
Lloyd, Wayne; Reese, Colin B.; Song, Quanlai; Vandersteen, Anthony M.; Visintin, Cristina; Zhang, Pei-Zhou
Journal of the Chemical Society, Perkin Transactions 1, 2000 , # 2 p. 165 - 176