3-氯-4-氨基苯硼酸频哪醇酯合成路线 （共 2 条）
反应条件
1: With potassium acetate in dimethyl sulfoxide 0.75 h; 2: With 1,1'-bis-(diphenylphosphino)ferrocene; (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride in dimethyl sulfoxide T=100°C; 4 h;
参考文献
BOEHRINGER INGELHEIM INTERNATIONAL GmbH; BOEHRINGER INGELHEIM PHARMA GmbH and CO KG
Patent: WO2005/118575 A1, 2005 ;
Location in patent: Page/Page column 80-81 ;
WO 2005/118575 A1
反应条件
1: With triethylamine in 1,4-dioxane 0.5 h; 2: With (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride in 1,4-dioxane; dichloromethane T=100°C; 20 h;
参考文献
X-CEPTOR THERAPEUTICS, INC.; SANKYO COMPANY, LIMITED
Patent: WO2004/58717 A1, 2004 ;
Location in patent: Page 80 ;
WO 2004/058717 A1
