反应条件
1: 12.93 g / methanol; dioxane / 2.5 h / Heating 2: 1.) H2, semicarbazide hydrochloride, NaOAc, 2.) 10percent aq. HCl, 36percent aq. CH2O / 1.) Raney Ni / 1.) EtOH, H2O, 50 psi, 2.) EtOH, H2O, heating, 30 min View Scheme
参考文献
European Journal of Medicinal Chemistry, , vol. 28, # 7-8 p. 601 - 608