反应条件
1: 1.) copper(I) iodide / 1.) Swern oxidation; 2.) THF, -78 deg C, dimethylsulfide 2: NaH / tetrahydrofuran; dimethylformamide 3: 1.) BH3; 2.) 30 percent H2O2, 12 percent NaOH / 1.) THF 4: mesyl chloride, triethylamine / CH2Cl2 View Scheme
参考文献
Chemical and pharmaceutical bulletin, , vol. 35, # 5 p. 2140 - 2143