反应条件
1: NaH / tetrahydrofuran; dimethylformamide 2: 1.) BH3; 2.) 30 percent H2O2, 12 percent NaOH / 1.) THF 3: mesyl chloride, triethylamine / CH2Cl2 4: H2, HCl / 10 percent Pd/C / ethanol View Scheme
参考文献
Chemical and pharmaceutical bulletin, , vol. 35, # 5 p. 2140 - 2143