反应条件
sodium hydride
1.) DMF, mineral oil, 5 deg C, 1 h, 2.) DMF, mineral oil, RT, 18 h; Yield given. Multistep reaction;
参考文献
Cross, Peter E.; Dickinson, Roger P.; Parry, M. John; Randall, Michael J.
Journal of Medicinal Chemistry, 1986 , vol. 29, # 3 p. 342 - 346