(8beta)-6-烯丙基麦角灵-8-羧酸甲酯合成路线 (共 11 条)
反应条件
1: With sodium hydroxide; water in methanol
T=20 - 30°C; 2 - 3 h;
2: With hydrogenchloride in methanol; water
T=0 - 5°C; pH=6 - 6.5; 1 - 2 h;
参考文献
Apotex Pharmachem Inc.
Patent: US2008/275240 A1, 2008 ;
Location in patent: Page/Page column 11-12 ;