反应条件
1.1: 1,4-diaza-bicyclo[2.2.2]octane / 1-methyl-pyrrolidin-2-one / 50 °C
1.2: 2.5 h / 50 °C
2.1: N,N-dimethyl acetamide / 2.67 h / 170 °C / |Sealed tube; |Microwave irradiation
View Scheme
参考文献
Moseley, Jonathan D.; Lenden, Philip; Lockwood, Mark; Ruda, Katinka; Sherlock, Jon-Paul; Thomson, Anthony D.; Gilday, John P.
Organic Process Research and Development, 2008 , vol. 12, # 1 p. 30 - 40